N-phosphorylation of pyrroles: An intramolecular migration reaction

Tasgin D. I., ÜNALEROĞLU C.

TETRAHEDRON LETTERS, vol.59, no.20, pp.1955-1957, 2018 (SCI-Expanded) identifier identifier

  • Publication Type: Article / Article
  • Volume: 59 Issue: 20
  • Publication Date: 2018
  • Doi Number: 10.1016/j.tetlet.2018.04.022
  • Journal Name: TETRAHEDRON LETTERS
  • Journal Indexes: Science Citation Index Expanded (SCI-EXPANDED), Scopus
  • Page Numbers: pp.1955-1957
  • Keywords: N-phosphorylation, Pyrrole, Intramolecular migration, Phosphonates, HETEROCYCLES, DERIVATIVES, ALKYLATION, BINDING, ACIDS
  • Hacettepe University Affiliated: Yes

Abstract

A new synthetic method is reported for the N-phosphorylation of pyrroles via intramolecular migration of a phosphonate diester group. The reaction proceeds under mild conditions and produces N-phosphorylated pyrrole derivatives in moderate to good yields. (C) 2018 Elsevier Ltd. All rights reserved.