N-phosphorylation of pyrroles: An intramolecular migration reaction

Tasgin D. I., ÜNALEROĞLU C.

TETRAHEDRON LETTERS, cilt.59, sa.20, ss.1955-1957, 2018 (SCI-Expanded) identifier identifier

  • Yayın Türü: Makale / Tam Makale
  • Cilt numarası: 59 Sayı: 20
  • Basım Tarihi: 2018
  • Doi Numarası: 10.1016/j.tetlet.2018.04.022
  • Dergi Adı: TETRAHEDRON LETTERS
  • Derginin Tarandığı İndeksler: Science Citation Index Expanded (SCI-EXPANDED), Scopus
  • Sayfa Sayıları: ss.1955-1957
  • Anahtar Kelimeler: N-phosphorylation, Pyrrole, Intramolecular migration, Phosphonates, HETEROCYCLES, DERIVATIVES, ALKYLATION, BINDING, ACIDS
  • Hacettepe Üniversitesi Adresli: Evet

Özet

A new synthetic method is reported for the N-phosphorylation of pyrroles via intramolecular migration of a phosphonate diester group. The reaction proceeds under mild conditions and produces N-phosphorylated pyrrole derivatives in moderate to good yields. (C) 2018 Elsevier Ltd. All rights reserved.